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STAT5b inhibitor 7

CAS No. 1818390-58-7

STAT5b inhibitor 7( Capstafin prodrug )

Catalog No. M12797 CAS No. 1818390-58-7

STAT5b inhibitor 7 (Capstafin prodrug) is the pivaloyloxymethyl ester prodrug of Capstafin.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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Biological Information

  • Product Name
    STAT5b inhibitor 7
  • Note
    Research use only, not for human use.
  • Brief Description
    STAT5b inhibitor 7 (Capstafin prodrug) is the pivaloyloxymethyl ester prodrug of Capstafin.
  • Description
    STAT5b inhibitor 7 (Capstafin prodrug) is the pivaloyloxymethyl ester prodrug of Capstafin, which is a potent, selective STAT5b inhibitor with Ki of 0.34 uM; inhibits STAT5b with selectivity over STAT5a in human tumor cells, inhibits cell viability and induces apoptosis in human tumor cells in a STAT5-dependent manner.
  • In Vitro
    ——
  • In Vivo
    ——
  • Synonyms
    Capstafin prodrug
  • Pathway
    JAK/STAT Signaling
  • Target
    STAT
  • Recptor
    STAT
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1818390-58-7
  • Formula Weight
    909.941
  • Molecular Formula
    C41H69NO17P2
  • Purity
    >98% (HPLC)
  • Solubility
    ——
  • SMILES
    CC(C)CCCCCCC(NCC1=CC=C(OP(OCOC(C(C)(C)C)=O)(OCOC(C(C)(C)C)=O)=O)C(OP(OCOC(C(C)(C)C)=O)(OCOC(C(C)(C)C)=O)=O)=C1)=O
  • Chemical Name
    ((((4-((8-methylnonanamido)methyl)-1,2-phenylene)bis(oxy))bis(oxo-l5-phosphanetriyl))tetrakis(oxy))tetrakis(methylene) tetrakis(2,2-dimethylpropanoate)

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Elumalai N, et al. ACS Chem Biol. 2015 Dec 18;10(12):2884-90.
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